121282-70-0Relevant articles and documents
A new facile method for the chemoselective reductive transformation of azides to N-(tert-butoxycarbonyl)amines
Kotsuki, Hiyoshizo,Ohishi, Takeshi,Araki, Tomohiro
, p. 2129 - 2132 (1997)
A new chemoselective procedure for the reductive transformation of organic azides to the corresponding N-(tert-butoxycarbonyl)amino derivatives using triethylsilane and di-tert-butyl dicarbonate in the presence of a catalytic amount of 20% Degussa Pd(OH)
COMPOUNDS, COMPOSITIONS AND METHODS FOR SYNTHESIS
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Paragraph 001588; 001589; 001590; 001591; 00756; 00757; 0076, (2019/01/10)
The present disclosure, among other things, provides technologies for synthesis, including reagents and methods for stereoselective synthesis. In some embodiments, the present disclosure provides compounds useful as chiral auxiliaries. In some embodiments, the present disclosure provides reagents and methods for oligonucleotide synthesis. In some embodiments, the present disclosure provides reagents and methods for chirally controlled preparation of oligonucleotides. In some embodiments, technologies of the present disclosure are particularly useful for constructing challenging internucleotidic linkages, providing high yields and stereoselectivity.
CYCLOHEXANEDIAMINE COMPOUNDS AND METHODS FOR THEIR PREPARATION
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, (2014/10/04)
The present invention provides processes for the preparation of cyclohexanediamine compounds of formula Ia and intermediates thereof. The compounds are useful as Syk kinase inhibitors and in various pharmaceutical compositions, and particularly useful for treating conditions mediated at least in part by Syk kinase activity.