13307-67-0Relevant articles and documents
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Kasparek,Heacock
, p. 2805,2808 (1966)
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A indole compound and its preparation method and application (by machine translation)
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Paragraph 0095; 0096; 0097, (2018/10/02)
The invention discloses a indole compound and its preparation method and application. The indole compounds of the structural formula such as formula (I) is shown. The indoles, rice galenical demonstrate the excellent inhibitory activity, the effect of most of the compound is obviously better than the positive control drug validamycin; especially compound I - 43, I - 44, I - 54, I - 73, II - 7 and II - 17, its galenical very good living body protection and treating effect, effect is better than the positive control; more specifically, compound I - 43 of the rice sheath blight bacteriostatic activity than validamycin activity is improved by nearly 300 times. The indole compounds in the prevention and/or treatment of rice sheath blight has great application prospects. In addition the compound of the invention is simple in construction, the preparation method is simple, and is suitable for large-scale industrial production. (I). (by machine translation)
N-carboxylated-2-substituted indoles and 2,3-disubstituted-2,3-dihydro-4- quinolones from 2- alkynylbenzamides
Okamoto, Noriko,Takeda, Kei,Yanada, Reiko
, p. 27 - 38 (2014/04/17)
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Chemoselective N-acylation of indoles and oxazolidinones with carbonylazoles
Heller, Stephen T.,Schultz, Erica E.,Sarpong, Richmond
supporting information; experimental part, p. 8304 - 8308 (2012/09/08)
Unique reactivity: In the presence of more reactive amine and alcohol functional groups and of carboxylic acids, the chemoselective N-acylation of indoles (see scheme) and oxazolidinones is achieved by taking advantage of the unique reactivity of carbonylazole acylating agents with catalytic amounts of 1,8-diazabicyclo[5.4.0]undec-7-ene (DBU). Copyright
