14338-21-7Relevant articles and documents
The inexpensive additive N-methylmorpholine effectively decreases the equivalents of nucleophiles in the catalytic highly enantioselective arylation of aryl aldehydes
Wang, Pei,Liu, Yue,Zhang, Ya-Lun,Da, Chao-Shan
supporting information, p. 443 - 450 (2017/07/25)
Highly enantioselective arylation of aryl aldehydes catalyzed by (S)-H8-BINOL-Ti(Oi-Pr)2 complex in the presence of N-methylmorpholine (NMM) as an effective and inexpensive additive is described for the first time. We found high enan
Sequential [3,3]-Sigmatropic Rearrangement/Nucleophilic Arylation of N -(Benzoyloxy)enamides towards the Preparation of Cyclic β-Aryl-β-amino Alcohols
Sato, Shohei,Takeda, Norihiko,Ueda, Masafumi,Miyata, Okiko
, p. 882 - 892 (2016/03/15)
A new method has been developed for the efficient synthesis of cyclic β-aryl-β-amino alcohol derivatives bearing a tetrasubstituted carbon center via the [3,3]-sigmatropic rearrangement of N-(benzoyl oxy)enamides followed by nucleophilic arylation reactio
Process for the Preparation of ?-C-Aryl Glucosides
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Paragraph 0356; 0357, (2014/05/20)
The present invention provides processes for stereoselectively preparing C-arylglucosides that can be useful as synthetic building block or drugs, including SGLT2 inhibitors.