15795-64-9Relevant academic research and scientific papers
ANTAGONISTS OF THE TOLL-LIKE RECEPTOR 1/2 COMPLEX
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Page/Page column 18; 19; 20; 21, (2014/02/16)
Provided are compounds, compositions and methods for treating Toll-like receptor 1/2 complex (TLRI/2) related inflammatory disorders. Small molecules, based on the benzotropolone scaffold, capable of influencing downstream signaling are dislcosed as well as methods of making and modifying these molecules. Also provided are methods for treating a subject for a clinical condition associated with Toll? like receptor complex 1/2 activation, comprising administering to the subject an effective amount of a benzotropolone compound.
Discovery of small-molecule inhibitors of the TLR1/TLR2 complex
Cheng, Kui,Wang, Xiaohui,Zhang, Shuting,Yin, Hang
supporting information, p. 12246 - 12249 (2013/02/23)
An important regulator of innate immunity, the protein complex of Toll-like receptors 1 and 2 (TLR1/TLR2) provides an attractive target for the treatment of various immune disorders. The novel compound CU-CPT22 can compete with the binding of the specific lipoprotein ligand to TLR1/TLR2 (see picture) with high inhibitory activity and specificity. Repression of downstream signaling from TNF-α and IL-1β was also observed. Copyright
