2127-09-5Relevant articles and documents
Peptide Tethering: Pocket-Directed Fragment Screening for Peptidomimetic Inhibitor Discovery
Arora, Paramjit S.,Marrone, Frank,Modell, Ashley E.,Panigrahi, Nihar R.,Zhang, Yingkai
supporting information, p. 1198 - 1204 (2022/02/05)
Constrained peptides have proven to be a rich source of ligands for protein surfaces, but are often limited in their binding potency. Deployment of nonnatural side chains that access unoccupied crevices on the receptor surface offers a potential avenue to
A coordinated synthesis and conjugation strategy for the preparation of homogeneous glycoconjugate vaccine candidates
Grayson, Elizabeth J.,Bernardes, Goncalo J. L.,Chalker, Justin M.,Boutureira, Omar,Koeppe, Julia R.,Davis, Benjamin G.
supporting information; experimental part, p. 4127 - 4132 (2011/07/07)
A sweet solution: A strategy for the synthesis of well-defined carbohydrate-based vaccines is presented. The approach couples complex oligosaccharide synthesis to site-specific conjugation methodology to provide pure glycoprotein vaccine candidates (see scheme). Copyright
Heteroaryl thioglycosides, a new class of substrates for glycosidases
Niemiec-Cyganek,Szeja
, p. 969 - 973 (2007/10/03)
We have found that heteroaryl thioglycosides are useful substrates of β-glucosidase from almond and can act as a new class of donors in transglycosylation reaction.
PYRANONE COMPOUNDS USEFUL TO TREAT RETROVIRAL INFECTIONS
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, (2008/06/13)
The present invention relates to compounds of formulae (I) and (II) which are pyran-2-ones, 5,6-dihydro-pyran-2-ones, 4-hydroxy-benzopyran-2-ones, 4-hydroxy-cycloalkyl[b]pyran-2-ones, and derivatives thereof, useful for inhibiting a retrovirus in a mammalian cell infected with said retrovirus, wherein R 10 and R 20 taken together are formulae (III) and (IV). STR1