Access to NH-aziridine-2-carboxamides through Davidsen acylimidodicarbonate activation

Add time:07/11/2019    Source:sciencedirect.com

Acylimidodicarbonates obtained from aziridine-2-carboxamides through Davidsen bis-Boc activation react with amine nucleophiles under mild conditions to form tertiary aziridine-2-carboxylic acid amides. NH aziridine-2-carboxylic acid amides were obtained by hydrogenolythic deprotection of N-Cbz derivatives.

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