Synthesis of 3-oxadiazolyl/triazolyl morpholines: Novel scaffolds for drug discovery

Add time:07/11/2019    Source:sciencedirect.com

Synthesis of isomeric 3-oxadiazolyl/triazolyl morpholines was performed based on a common intermediate on the gram scale. The target compounds were designed as novel scaffolds for the medicinal chemistry. The key reaction was an electrochemical CH-oxidation of N-Boc morpholine.

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