2H-Pyran-2-ones as synthons for (E)-α,β-didehydroamino acid derivatives

Add time:08/04/2019    Source:sciencedirect.com

2H-Pyran-2-ones with the defined (E)-structure of a α,β-didehydroamino acid unit were used as synthons for a series of configurationally stable (E)-α,β-didehydroamino acid derivatives containing a benzoyl protected amino function and a pyrazolyl residue. They were derived from 2H-pyran-2-ones and hydrazines under various reaction conditions. A possibility of the formation of (Z)-isomers from the above-mentioned precursors is also discussed.

We also recommend Trading Suppliers and Manufacturers of (4-CHLORO-BENZOYLAMINO)-ACETIC ACID (cas 13450-77-6). Pls Click Website Link as below: cas 13450-77-6 suppliers

Prev:Anthranilic acid based CCK1 antagonists: the 2-indole moiety may represent a “needle” according to the recent homonymous concept
Next:Anthranilic acid derivatives: a new class of non-peptide CCK1 receptor antagonists)