190792-74-6

Basic information

• Product Name: (3S,4S)-N-Boc-3-amino-4-hydroxypyrrolidine
• Synonyms: (3s,4s)-n-boc-3-amino-4-hydroxypyrrolidine;1-Pyrrolidinecarboxylicacid,3-amino-4-hydroxy-,1,1-dimethylethylester,(3S,4S)-(9CI);(3S,4S)-3-Amino-4-hydroxypyrrolidine-1-carboxylic acid tert-butyl ester;(3S,4S)-tert-Butyl 3-amino-4-hydroxypyrrolidine-1-carboxylate;1-Boc-(3S,4S)-3-aMino-4-hydroxypyrrolidine;(3S,4S)-4-aMino-1-N-tert-butyloxycarbonyl-3-hydroxypyrrolidine;Trans-(3S,4S)-1-Boc-3-aMino-4-hydroxypyrrolidine;tert-butyl (3S,4S)-3-amino-4-hydroxypyrrolidine-1-carboxylate
• CAS NO: 190792-74-6
• Molecular Formula: C₉H₁₈N₂O₃
• Molecular Weight: 202.25
• Product Categories: AMINOACID
• Mol File: 190792-74-6.mol

Chemical Properties

• Boiling Point: 308.762 °C at 760 mmHg
• Flash Point: 140.535 °C
• Appearance: /
• Density: 1.179
• Storage Temp.: 2-8°C(protect from light)
• PKA: 14.36±0.40(Predicted)
• CAS DataBase Reference: (3S,4S)-N-Boc-3-amino-4-hydroxypyrrolidine(CAS DataBase Reference)
• NIST Chemistry Reference: (3S,4S)-N-Boc-3-amino-4-hydroxypyrrolidine(190792-74-6)
• EPA Substance Registry System: (3S,4S)-N-Boc-3-amino-4-hydroxypyrrolidine(190792-74-6)

Safety Data

• Hazardous Substances Data: 190792-74-6(Hazardous Substances Data)

Usage

Uses

Used in Pharmaceutical Development:
(3S,4S)-N-Boc-3-amino-4-hydroxypyrrolidine is used as an intermediate compound in the synthesis of various pharmaceuticals. Its unique stereochemistry and the presence of the Boc protecting group make it a valuable building block for the development of new drugs.
Used in Scientific Research:
In the field of scientific research, (3S,4S)-N-Boc-3-amino-4-hydroxypyrrolidine serves as a key compound for studying the properties and reactivity of Pyrrolidine derivatives. Its use in research helps in understanding the potential applications and limitations of this class of compounds in various chemical and biological processes.
Used in Chemical Synthesis:
(3S,4S)-N-Boc-3-amino-4-hydroxypyrrolidine is used as a protected amino alcohol in the synthesis of complex organic molecules. The Boc protecting group allows for selective reactions to occur at other sites on the molecule, while the amino and hydroxy groups remain protected from unwanted side reactions. This makes it a useful tool in the synthesis of a wide range of chemical products.

Upstream product

• 203434-45-1 (±)-tert-butyl 3-azido-4-hydroxypyrrolidine-1-carboxylate 
• 252574-03-1 (3S,4S)-1-tert-butoxycarbonyl-trans-3-benzylamino-4-hydroxypyrrolidine 
• 4248-19-5 tert-butyl carbazate 
• 24424-99-5 di-tert-butyl dicarbonate 
• 73286-70-1 N-(tert-butoxycarbonyl)-3-pyrroline 
• 114214-49-2 1-tert-butoxycarbonyl-3,4-epoxypyrrolidine 
• 252574-02-0 (±)-trans-tert-butyl 3-bromo-4-hydroxypyrrolidine-1-carboxylate 
• 926913-20-4 (3R,4S)-1-N-tert-butyloxycarbonyl-4-(4,4'-dimethoxytrityloxy)-3-mesyloxy-pyrrolidine 
• 183184-52-3 1-((3S,4S)-3-azido-4-hydroxypyrrolidin-1-yl)-2,2,2-trifluoroethan-1-one 
• 164931-85-5 meso-N-trifluoroacetyl-3-pyrroline oxide 
• 1202067-33-1 (3S,4S)-3-azido-4-(trimethylsilanyloxy)pyrrolidine-1-carboxylic acid tert-butyl ester 
• 190792-84-8 (3S,4S)-3-azido-4-hydroxy-pyrrolidine-1-carboxylic acid tert-butyl ester 

Downstream Products

• 1333414-02-0 (3S,4S)-tert-butyl 3-(tert-butyldiphenylsilyloxy)-4-(trifluoromethylsulfonamido)pyrrolidine-1-carboxylate 
• 1215210-04-0 (3S,4S)-3-amino-4-hydroxypyrrolidine dihydrochloride 
• 1202067-40-0 (3S,4S)-3-benzoylamino-4-hydroxypyrrolidine-1-carboxylic acid tert-butyl ester 
• 138026-97-8 (3R,4S)-4-amino-1-N-tert-butyloxycarbonyl-3-hydroxypyrrolidine 
• 859213-33-5 (3S,4S)-tert-butyl 3-(dimethyl amino)-4-hydroxypyrrolidine-1-carboxylate 
• 1202067-41-1 (3aS,6aR)-2-phenyl-3a,4,6,6a-tetrahydropyrrolo[3,4-d]oxazole-5-carboxylic acid tert-butyl ester 

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