Xanthine Functionalized Congeners as Potent Ligands at A2-Adenosine Receptors

DOI: 10.1021/jm00384a037

Source and publish data:

Journal of Medicinal Chemistry p. 211 - 214 (1987)

Update date:2022-08-05

Topics:

Authors:

Jacobson, Kenneth A.

Ukena, Dieter

Padgett, William

Daly, John W.

Kirk, Kenneth L.

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Article abstract of DOI:10.1021/jm00384a037

Amide derivatives of a carboxylic acid congener of 1,3-dialkylxanthine, having a 4-<(carboxymethyl)oxy>phenyl substituent at the 8-position, have been synthesized in order to identify potent antagonists at A₂-adenosine receptors stimulatory to

Full text of DOI:10.1021/jm00384a037

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