Structure-activity relationships of cyclic opioid peptide analogues containing a phenylalanine residue in the 3-position

DOI: 10.1021/jm00394a027

Source and publish data:

Journal of Medicinal Chemistry p. 2094 - 2099 (1987)

Update date:2022-08-05

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Authors:

Schiller

Nguyen Nguyen

Maziak Maziak

Wilkes Wilkes

Lemieux Lemieux

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Article abstract of DOI:10.1021/jm00394a027

Ten analogues of the highly μ-receptor selective cyclic opioid peptide H-Tyr-D-Orn-Phe-Asp-NH₂ (1) were synthesized by the solid-phase method and were characterized in vitro in μ- and δ-receptor representative binding assays and bioassays. Thes

Full text of DOI:10.1021/jm00394a027

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