C-Alkylation of Phenylthio Aziridine Carbonylates

DOI: 10.1246/cl.1987.49

Source and publish data:

Chemistry Letters p. 49 - 52 (1987)

Update date:2022-08-03

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Authors:

Seebach, Dieter

Haner, Robert

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Article abstract of DOI:10.1246/cl.1987.49

The N-t-butyl and N-benzyl aziridine carboxylic acid phenylthiol esters are deprotonated in the α-carbonyl position and alkylated by alkyl halides, by aldehydes, and by nitrostyrene.The diastereselectivities in the additions to trigonal centers range from

Full text of DOI:10.1246/cl.1987.49

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