Tetrahedron Letters p. 401 - 404 (1987)
Update date:2022-07-30
Topics: Reactif
Galzi, J. L.
Ilien, B.
Simon, E. J.
Goeldner, M.
Hirth, C.
The synthesis of several fentanyl derivatives is reported.The binding affinity of these compounds to membrane opioid receptors is also presented.Several potentially irreversible aryldiazonium ligands were tested for irreversible inactivation of opioid receptors.Compound 13 was shown to inactivate up to 50percent of rat brain opioid receptors, in a ligand-protectable manner.It is therefore a potentially efficient affinity probe for these receptors.
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