AMINO-ALCOHOL DIPEPTIDE ANALOGUES: A SIMPLE SYNTHESIS OF A VERSATILE ISOSTERE FOR THE DEVELOPMENT OF PROTEINASE INHIBITORS

DOI: 10.1016/S0040-4039(00)96784-4

Source and publish data:

Tetrahedron Letters p. 5569 - 5572 (1987)

Update date:2022-08-04

Topics:

Authors:

Arrowsmith, R. J.

Davies, D. E.

Fogden, Y. C.

Harris, C. J.

Thompson, C.

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Article abstract of DOI:10.1016/S0040-4039(00)96784-4

Two simple approaches to an amino-alcohol isostere of proteolytically-cleavable dipeptide sequences are described; this isostere is incorporated into stereochemically-defined tetrapeptide analogues.

Full text of DOI:10.1016/S0040-4039(00)96784-4

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