Aromatase inhibitors: Synthesis, biological activity, and structure of 1,2-imidazolylmethylcyclopentanol derivatives

DOI: 10.1248/cpb.43.2152

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 2152 - 2158 (1995)

Update date:2022-08-02

Topics:

Authors:

Kato Kato

Ikeda Ikeda

Sugita Sugita

Nitta Nitta

Enari Enari

Kashima Kashima

Konno Konno

Niimura Niimura

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1248/cpb.43.2152

Two series of 1,2-disubstituted imidazolylmethylcyclopentanol derivatives (5a-d, 10a-d) were prepared by using easily available methyl 2- oxocyclopentanecarboxylate as the starting material. Evaluation of the aromatase inhibitory activities in vitro was p

Full text of DOI:10.1248/cpb.43.2152

NII-Electronic Library Service

Products guided by the article

Product name:1-[(4-chlorophenyl)methyl]-2-oxocyclopentanecarboxylic acid methyl ester

Cas No:115851-73-5

R&D Labs maybe for 115851-73-5

Zhonghao (dalian) Research and Design Institute of Chemical Industry Co., Ltd

Contact:+86 411 84674606

Address:201, Huangpu Road , Shahekou District, Dalian ,116023-China
Shijiazhuang Haotian Chemical Co., Ltd.

Contact:86-311-85044374

Address:293 Donggang Road
NINGBO PANGS CHEM INT’L CO.,LTD.

Contact:+86-574-27666845

Address:FLOOR 21,BUILDING NO.11,XIN TIAN DI,NO.689 SHI JI ROAD,NINGBO CHINA
Dalian Synco Chemical Co., Ltd.

Contact:+86-411-83635150

Address:Rm 1004, 24, Tangshan Street, Dalian
Maithili Life Sciences

Contact:+91 9963263336

Address:Plot#146A, IDA Mallapur, Hyderabad - 500072

Relevant to this article

Gold(I)-catalyzed arylmethylation of terminal alkynes

Doi:10.1016/j.tetlet.2009.03.067
(2009)
Efficient synthesis of aminomethylated pyrroloindoles and dipyrrolopyridines via controlled copper-catalyzed domino multicomponent coupling and bis-cyclization

Doi:10.1021/jo900681p
(2009)
Molecular recognition in anisotropic media. Binding of alkylpyridines to amphiphilic zinc porphyrins incorporated in liposomal bilayer membranes

Doi:10.1039/b817241b
(2009)
Cobaloximes with bis(thiophenyl)glyoxime: Synthesis and structure - Property relationship study

Doi:10.1021/om900065k
(2009)
Synthetically useful Bronsted acid-promoted arylbenzyl ether → o-benzylphenol rearrangements

Doi:10.1021/jo9007833
(2009)
Synthesis of (3,5-aryl/methyl-1H-pyrazol-1-yl)-(5-arylamino-2H-1,2,3- triazol-4-yl)methanone

Doi:10.1002/jccs.200800114
(2008)

Article Doi