
Journal of Medicinal Chemistry p. 2081 - 2086 (1988)
Update date:2022-08-04
Topics:
Van Dort
Ciliax
Gildersleeve
Sherman
Rosenspire
Young
Junck
Wieland
Two isomeric iodinated analogues of the peripheral benzodiazepines binding site (PBS) ligand Ro5-4864 have been synthesized and labeled in high specific activity with iodine-125. Competitive binding assays conducted with the unlabeled analogues indicate h
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