A PROSTHETIC GROUP FOR THE RAPID INTRODUCTION OF FLUORINE INTO PEPTIDES AND FUNCTIONALIZED DRUGS

DOI: 10.1016/S0022-1139(00)81606-1

Source and publish data:

Journal of Fluorine Chemistry p. 339 - 348 (1988)

Update date:2022-07-31

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Authors:

Jacobson, Kenneth A.

Furlano, David C.

Kirk, Kenneth L.

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Article abstract of DOI:10.1016/S0022-1139(00)81606-1

Fluoride ion as the tetrabutylammonium salt displaces bromide in para-substituted benzyl bromides in acetonitrile or dimethylformamide.The p-bromomethyl benzoyl (BMB) group has been coupled to amino groups, including peptide amino groups, via its N-hydrox

Full text of DOI:10.1016/S0022-1139(00)81606-1

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