Asymmetric Allylic Amination of Morita-Baylis-Hillman Adducts with Simple Aromatic Amines by Nucleophilic Amine Catalysis

DOI: 10.1055/s-0037-1611740

Source and publish data:

Synlett p. 703 - 708 (2019)

Update date:2022-08-04

Topics:

Authors:

Zhao, Shuai

Chen, Zhi-Li

Rui, Xue

Gao, Ming-Mei

Chen, Xin

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Article abstract of DOI:10.1055/s-0037-1611740

Asymmetric allylic amination of Morita-Baylis-Hillman (MBH) adducts with simple aromatic amines is successfully realized by nucleophilic amine catalysis. A range of substituted α-methylene-β-arylamino esters is accessed in moderate to high yields (up to 8

Full text of DOI:10.1055/s-0037-1611740

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