C-GLYCOSYLATION OF SUBSTITUTED HETEROCYCLES UNDER FRIEDEL-CRAFTS CONDITIONS (I): A TWO-STEP SYNTHESIS OF THE THIENOPYRIMIDINE c-NUCLEOSIDE ANALOG OF INOSINE.

DOI: 10.1016/0040-4039(88)85286-9

Source and publish data:

Tetrahedron Letters p. 3537 - 3540 (1988)

Update date:2022-08-05

Topics:

Authors:

Rao, Sunkada P.

Rao, Kambhampati V. B.

Otter, Brian A.

Klein, Robert S.

Ren, Wu-Yun

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Article abstract of DOI:10.1016/0040-4039(88)85286-9

Direct stannic chloride catalyzed C-glycosylation of N-formyl-4-amino-3-carboalkoxy thiophenes with 1-O-acetyl-O-benzoyl-β-D-ribofuranose, followed by annelation of a fused pyrimidone ring upon treatment with ammonia, constitutes a short approach to the synthesis of a new C-nucleoside inosine analog.

Full text of DOI:10.1016/0040-4039(88)85286-9

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