Concise synthesis of pyrimido-azocine derivatives via aza-claisen rearrangement and intramolecular heck reaction

DOI: 10.1055/s-0029-1219276

Source and publish data:

Synthesis p. 1315 - 1320 (2010)

Update date:2022-08-03

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Authors:

Majumdar

Mondal, Shovan

Ghosh, Debankan

Chattopadhyay, Buddhadeb

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Article abstract of DOI:10.1055/s-0029-1219276

An expedient approach involving BF₃OEt₂-catalyzed aza-Claisen rearrangement and palladium-catalyzed intramolecular Heck reaction for the synthesis of pyrimidine-fused azocine derivatives is described. The mechanistic interpretation o

Full text of DOI:10.1055/s-0029-1219276

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