Tetrahedron Letters p. 1053 - 1056 (2011)
Update date:2022-08-04
Topics:
Pham, Helen Trinh
Hanson, Robert N.
Olmsted, Sandra L.
Kozhushnyan, Anton
Visentin, Adam
Weglinsky, Paul J.
Massero, Chris
Bailey, Kristen
The preparation of the novel isomeric 6- and 7-propargyloxy derivatives of 4-(3-fluoroanilino)-quinazoline was achieved using a six-step process. An alternate method to the 7-propargyloxy derivative and analogous 7-propargyloxy containing compounds is als
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