A practical approach to Dideoxy-1,4- and 1,5-iminopentitols from protected sugar hemiacetals

Article abstract of DOI:10.1016/j.carres.2019.107855

The convenient and straightforward preparation of dideoxy-1,4- and 1,5-iminopentitol derivatives from protected sugar hemiacetals by way of N-tert-butanesulfinyl glycosylamines and open-chain aminoalditols is reported. The synthetic procedure is a method of choice for the making of these important scaffolds of biological interest.