Nucleophilic ring opening of C2-symmetric aziridines. Synthetic equivalents for the β-cation of aspartic acid

DOI: 10.1016/S0040-4039(00)98816-6

Source and publish data:

Tetrahedron Letters p. 1903 - 1906 (1990)

Update date:2022-08-05

Topics:

Authors:

Tanner Tanner

Birgersson

Dhaliwal

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Article abstract of DOI:10.1016/S0040-4039(00)98816-6

The non-racemic C₂-symmetric aziridines 7 and 8, easily available from (+)- and (-)-tartaric acid, respectively, undergo rapid nucleophilic attack to yield products formally derived from the β-cation of L- or D-aspartic acid.

Full text of DOI:10.1016/S0040-4039(00)98816-6

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