Bioorganic and Medicinal Chemistry Letters p. 760 - 763 (2011)
Update date:2022-08-02
Topics:
Nagasawa, Johnny Y.
Song, Jenny
Chen, Huanming
Kim, Hong-Woo
Blazel, Julie
Ouk, Samedy
Groschel, Bettina
Borges, Virginia
Ong, Voon
Yeh, Li-Tain
Girardet, Jean-Luc
Vernier, Jean-Michel
Raney, Anneke K.
Pinkerton, Anthony B.
SAR studies on the quinolone carboxylic acid class of HIV-1 integrase inhibitors focused on improving the metabolic stability and led to the discovery of 27 and 38.
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