Synthesis of Leu-Abu(P) and Glu-Abu( P)-Leu. Isosteres of ser(P)-peptides

DOI: 10.1016/S0040-4039(00)97464-1

Source and publish data:

Tetrahedron Letters p. 3759 - 3762 (1990)

Update date:2022-08-04

Topics:

Authors:

Tong Tong

Perich Perich

Johns Johns

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0040-4039(00)97464-1

Boc-Asp-O₁-Bu was efficiently converted to Boc-Abu(PO₃Me₂)-O₁-Bu in five steps then to Boc-Abu(PO₃Me₂)OH in two steps. Both the protected amino acids were used in the syntheses of Boc-Leu-A

Full text of DOI:10.1016/S0040-4039(00)97464-1

Products guided by the article

Product name:L-Leucine, N-[(1,1-dimethylethoxy)carbonyl]-L-a-glutamyl-4-(dimethoxyphosphinyl)- L-2-aminobutanoyl-, bis(phenylmethyl) ester

Cas No:130568-17-1

R&D Labs maybe for 130568-17-1

Guangzhou PI & PI Biotech Inc. Ltd.

Contact:+86-20-81716320

Address:13th Floor, Xinbao Technology Industrial Park, No. 2 Ruixiang Road, Huangpu District, Guangzhou,Guangdong,China
HANGZHOU TOYOND BIOTECH CO., LTD

Contact:+86-571-86965177

Address:No. 189, Fengqi East Road, Hangzhou, China
zhengzhou Triz Pharma-Tech Co., Ltd

website:http://www.Trizpharma-tech.com

Contact:+86-0371-86597269，53392065

Address:High-tech Industrial Development Zone, Zhengzhou City, NO.7 Holly Street
Linyi Shengxin Pharmaceutical R&D Co., Ltd

Contact:+86-18653953873

Address:West First of Yufeng Road, Yishui County
Guangxi Nanning Guangtai Agriculture Chemical Co.,Ltd

Contact:+86-771-2311266

Address:Room703,Building12, Software Park Phase II,NO.68,Keyuan Road,Nanning City,Guangxi,China

Relevant to this article

An efficient convergent access to spiroketal segment of (+)-spiroxaline methyl ether

Doi:10.1055/s-0030-1258456
(2011)
Direct Nucleophilic Difluoromethylation of Carbonyl Compounds

Doi:10.1021/acs.orglett.6b01425
(2016)
Magnetic Field Effects and Reaction Mechanism in Photoredox Reaction of Nitro Group

Doi:10.1246/cl.1990.1559
(1990)
Iridium(I)-catalysed tandem hydrosilylation-protodesilylation of imines

Doi:10.1002/ejoc.200500168
(2005)
Doi:10.1016/S0040-4039(01)97652-X
(1969)
Straightforward preparation of functionalized α-CF ₂-galactosides through an oxygen to carbon acyl migration

Doi:10.1002/chem.201100183
(2011)

Article Doi