Directed lithiation of 3,5-dichloroaniline and its application in the synthesis of 1,3-dichloro-6,7,8,9,10,12-hexahydroazepino[2,1-b][5- 14C]quinazoline monohydrochloride

DOI: 10.1002/jlcr.2580340603

Source and publish data:

Journal of labelled compounds and radiopharmaceuticals p. 505 - 512 (1994)

Update date:2022-08-06

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Authors:

Ekhato Ekhato

Huang Huang

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Article abstract of DOI:10.1002/jlcr.2580340603

1,3-Dichloro-6,7,8,9,10,12-hexahydroazepino[2,1-b][5-¹⁴C]quinazoline monohydrochloride (1) was synthesized in 12% overall yield starting from 3,5- dichloroaniline, and a radiochemical purity of 99.6% was obtained. The synthetic sequence was fac

Full text of DOI:10.1002/jlcr.2580340603

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