Synthesis of 3-carbamoylecgonine methyl ester analogues as inhibitors of cocaine binding and dopamine uptake

DOI: 10.1021/jm00106a035

Source and publish data:

Journal of Medicinal Chemistry p. 702 - 705 (1991)

Update date:2022-09-26

Topics:

Authors:

Kline Jr.

Wright Wright

Eshleman

Fox Fox

Eldefrawi

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Article abstract of DOI:10.1021/jm00106a035

Five (1R-2-exo-3-exo)-3-(N-phenylcarbamoyl)ecgonine methyl ester analogues were synthesized and characterized by ¹H and ¹³C NMR, IR, and thermospray MS. The compounds were synthesized in two or three steps as (-)-stereoisomers from (

Full text of DOI:10.1021/jm00106a035

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