Electrophilic cyclizations of 2-fluoroalk-3-yn-1-ones: Room-temperature synthesis of diversely 2,5-disubstituted 3,4-fluorohalofurans

DOI: 10.1002/ejoc.201100344

Source and publish data:

European Journal of Organic Chemistry p. 2767 - 2771 (2011)

Update date:2022-08-02

Topics:

Authors:

Li, Yan Li, Yan

Wheeler, Kraig A.

Dembinski, Roman

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1002/ejoc.201100344

A 5-endo-dig halocyclization of 2-fluoroalk-3-yn-1-ones with the use of N-iodo- and N-bromosuccinimide, in the presence of gold chloride/zinc bromide (5:20 mol-%, dichloromethane), under ambient conditions, provides a facile method for the synthesis of 2,

Full text of DOI:10.1002/ejoc.201100344

Products guided by the article

Product name:3-bromo-4-fluoro-2-(4-methylphenyl)-5-phenylfuran

Cas No:1310738-68-1

R&D Labs maybe for 1310738-68-1

Chengdu King-tiger Pharm-chem. Tech. Co., Ltd

Contact:028-85317716

Address:Tianfu Life Science Park, No. 88 South Keyuan Road, Gaoxin District, Chengdu City, Sichuan Province, PRC.
SunaTech Inc.

Contact:+86 512 6287 2180

Address:398 Ruoshui Road, Suzhou Industrial Park, Suzhou, Jiangsu, P. R. China
lianyungang jinkang pharmaceutical technology co., ltd.

Contact:008651885445517

Address:Jinshan industrial park, Ganyu county, Lianyungang, Jiangsu Province, 222115, China
Anhui Xinyuan Technology Co.,Ltd

Contact:0086-559-3515800

Address:No.16 Zijin Rd, Circular Economic Zone, Huizhou District, Huangshan Anhui China
Hangzhou Chemfar Ltd.

Contact:+86-571-87859231, 87859237, 87859239

Address:1606,Huarong Times Mansion, No.3880 Jiangnan Avenue, Binjiang District, Hangzhou, China, 310053

Relevant to this article

A practical strategy for the structural diversification of aliphatic scaffolds through the palladium-catalyzed picolinamide-directed remote functionalization of unactivated C(sp³)-H bonds

Doi:10.1002/anie.201100984
(2011)
Synthesis and structure-activity relationship for new series of 4-phenoxyquinoline derivatives as specific inhibitors of platelet-derived growth factor receptor tyrosine kinase

Doi:10.1016/j.bmc.2003.08.020
(2003)
A highly effective phosphinite ligand derived from D-mannitol for Rh- catalyzed asymmetric hydrogenation

Doi:10.1016/S0040-4039(98)02457-5
(1999)
Doi:10.1021/ic50202a058
(1979)
Reductive-alkylation and aromatic coupling reactions of 1,4-benzoquinone derivatives promoted by ethylaluminum dichloride

Doi:10.1016/S0022-328X(98)00865-1
(1998)
Doi:10.1246/bcsj.50.1097
(1977)

Article Doi