Synthesis and screening of (E)-1-(β-D-galactopyranosyl)-4-(aryl)but-3- ene-2-one against Mycobacterium tuberculosis

DOI: 10.1016/j.bmcl.2011.05.037

Source and publish data:

Bioorganic and Medicinal Chemistry Letters p. 3947 - 3950 (2011)

Update date:2022-08-03

Topics:

Authors:

Mugunthan

Ramakrishna, Kuppala

Sriram, Dharmarajan

Yogeeswari, Perumal

Ravindranathan Kartha

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/j.bmcl.2011.05.037

A series of galactose-derived aryl enones were synthesised and screened against Mycobacterium tuberculosis H₃₇Rv. Preliminary results were promising with MIC values in the range 1.56-12.5 μg/mL.

Full text of DOI:10.1016/j.bmcl.2011.05.037

Products guided by the article

Product name:C₁₉H₂₆O₉

Cas No:1314797-70-0

R&D Labs maybe for 1314797-70-0

JenKem Technology Co., Ltd.

Contact:86-10-62983737; +86-10-51287608

Address:4/F Building C, 2 Shangdi Xinxi Road
Heliosense Biotechnologies, Inc.

Contact:+86-592-5667290

Address:Xiamen Torch Hi-tech Zone Venture Weiye Building S506
Zhengzhou Xinlian Chemical Tech Co. ,Ltd

Contact:0371-65771781 021-52042910

Address:H Part, Building I, No. 700 Gonglu Road, Pudong New Area, Shanghai
Sigma-Aldrich Chemie GmbH

website:http://www.sigmaaldrich.com

Contact:800 558-9160

Address:Industriestrasse 25CH-9471 Buchs SGSwitzerland
Suzhou CarbonWell Pharma-Tech Co., Ltd

Contact:Tel: + 86 (0)512-8898-1216; + 86-18606258602

Address:2358 Changan Road, Wujiang Scientific Innovation Park, Wujiang, Jiangsu Province, P. R. China 215200

Relevant to this article

Concise synthesis of the antidepressive drug candidate GSK1360707 by a highly enantioselective gold-catalyzed enyne cycloisomerization reaction

Doi:10.1002/chem.201101346
(2011)
Synthesis of 7α,12α-dihydroxy-3α-[2-(β-D-glucopyranosyl)acetyl]- 5β-cholan-24-oic acid

Doi:10.1016/0039-128X(90)90033-8
(1990)
Cp₂ZrCl₂-Catalyzed cycloalumination of acetylenic alcohols and propargylamines by Et₃Al

Doi:10.1007/s11172-011-0013-2
(2011)
Amino-acids and peptides. XXIV. The use of esters of 1-hydroxypiperidine and of other NN-dialkylhydroxylamines in peptide synthesis and as selective acylating agents.

Doi:10.1039/jr9650006814
(1965)
Synthesis and biological evaluation of triazolyl 13α-estrone-nucleoside bioconjugates

Doi:10.3390/molecules21091212
(2016)
Synthesis and crystal structures of [CuCl₂(μ-NSPh₃)]₂ and [CuCl₂(Ph₃SN)₂]: Novel copper complexes bearing organic λ⁶-sulfanenitrile as ligand

Doi:10.1246/cl.2002.1000
(2002)

Article Doi