Synthesis and Some Pharmacological Properties of Potent and Selective Antagonists of the Vasopressor (V1-Receptor) Response to Arginine-Vasopressin

DOI: 10.1021/jm00080a027

Source and publish data:

Journal of Medicinal Chemistry p. 382 - 388 (1992)

Update date:2022-09-26

Topics:

Authors:

Manning, Maurice

Stoev, Stoytcho

Bankowski, Krzysztof

Misicka, Aleksandra

Lammek, Bernard

et al. et al.

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1021/jm00080a027

We report the solid-phase synthesis of eight position-9-modified analogues of the potent V₁-receptor antagonist of arginine-vasopressin, <1-(β-mercapto-β,β-pentamethylenepropionic acid),2-O-methyltyrosine>arginine-vasopressin (d(CH2)5Tyr(Me)AVP

Full text of DOI:10.1021/jm00080a027

Products guided by the article

Product name:<β-(benzylthio)-β,β-pentamethylenepropionyl>-Tyr(Me)-Phe-Gln-Asn-Cys(Bzl)-Pro-Arg(Tos)-Val-NH2

Cas No:133201-31-7

R&D Labs maybe for 133201-31-7

Luoyang Aoda chemical Co.,Ltd.

Contact:+86-379-67518785 67516588

Address:MiaoWan industry district,YanShi City,Henan,China
Molobelamltrading

Contact:27-792-602929

Address:SIDNEY MUFAMADI STREET 009949 X44 0700 POLOKWANE,LIMPOPO
Synchemie Co., Ltd.

website:http://www.synchemie.com/

Contact:+86-574-87642758

Address:Room 901, Yinyi Bund Building， 132 Renmin Road
Anyang Double Circle Auxiliary CO.,LTD

Contact:0086-134 6082 4403

Address:dongfeng road, anyang city, henan province,china
Zhenjiang Haitong Chemical Industry Co., Ltd.

Contact:+86 (511) 8448-0369

Address:Baoyan Town, Dantu District, Zhenjiang City, Jiangsu, China

Relevant to this article

Surface active benzodiazepine-bromo-alkyl conjugate for potential GABA _A-receptor purification

Doi:10.1039/c1ob05210a
(2011)
Sodium hydride induced N-arylation of diisopropyl azodicarboxylate by aryl trifluoromethanesulfonates

Doi:10.1055/s-0034-1380143
(2015)
Synthesis and characterization of biologically active new Schiff bases containing 3-functionalized 1,2,4-triazoles and their zinc(II) complexes: Crystal structure of 4-bromo-2-[(E)-(1H-1,2,4-triazol-3-ylimino)- methyl]phenol

Doi:10.1002/aoc.1833
(2011)
(Dicyanoiodo)benzene - A stable tricoordinate iodine(III) compound with three carbon ligands

Doi:10.1016/S0040-4039(00)74870-2
(1991)
Pd/Cu-cocatalyzed reigoselective arylation of thiazole derivatives at 2-position under ligand-free conditions

Doi:10.1039/c5ra08703a
(2015)
Naphthopyranone glycosides from Paepalanthus bromelioides

Doi:10.1016/S0031-9422(97)00952-7
(1998)

Article Doi