Synthesis and Some Pharmacological Properties of Potent and Selective Antagonists of the Vasopressor (V1-Receptor) Response to Arginine-Vasopressin

DOI: 10.1021/jm00080a027

Source and publish data:

Journal of Medicinal Chemistry p. 382 - 388 (1992)

Update date:2022-09-26

Topics:

Authors:

Manning, Maurice

Stoev, Stoytcho

Bankowski, Krzysztof

Misicka, Aleksandra

Lammek, Bernard

et al. et al.

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Article abstract of DOI:10.1021/jm00080a027

We report the solid-phase synthesis of eight position-9-modified analogues of the potent V₁-receptor antagonist of arginine-vasopressin, <1-(β-mercapto-β,β-pentamethylenepropionic acid),2-O-methyltyrosine>arginine-vasopressin (d(CH2)5Tyr(Me)AVP

Full text of DOI:10.1021/jm00080a027

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