Amide Bond Replacements: Incorporation of a 2,5,5-Trisubstituted Imidazoline into Dipeptides and into a CCK-4 Derivative.

DOI: 10.1016/S0040-4039(00)79701-2

Source and publish data:

Tetrahedron Letters p. 2277 - 2280 (1991)

Update date:2022-08-02

Topics:

Authors:

Gilbert, Ian

Rees, David C.

Richardson, Reginald S.

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Article abstract of DOI:10.1016/S0040-4039(00)79701-2

Synthetic methodology for the introduction of a 2,5,5-trisubstituted imidazoline ring as an amide replacement into dipeptide derivatives of Phe, Trp, Lys(N⁶-CBZ) and Nle is described.This replacement is also incorporated into the Trp-Nle bond o

Full text of DOI:10.1016/S0040-4039(00)79701-2

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