The synthesis of 7-alkoxyindoles

Article abstract of DOI:10.1080/00397919108020827

A number of protected 7-hydroxyindoles was prepared by reaction of the protected 2-nitrophenols with vinylmagnesium bromide. Benzhydryl was shown to be the protecting group of choice, giving good yields of the indole and being readily removed for subsequent transformations of the 7-hydroxy function.

Full text of DOI:10.1080/00397919108020827

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Synthetic Communications: An
International Journal for Rapid
Communication of Synthetic
Organic Chemistry
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The Synthesis of 7-
Alkoxyindoles
David Dobson a , Alec Todd a & Jeremy Gilmore a
a Chemistry Department , Eli Lilly and Co. Ltd., Lilly
Research Centre Ltd. , Erl Wood Manor, Windlesham,
Surrey, GU20 6PH, England
Published online: 23 Sep 2006.
To cite this article: David Dobson , Alec Todd & Jeremy Gilmore (1991) The
Synthesis of 7-Alkoxyindoles, Synthetic Communications: An International Journal
for Rapid Communication of Synthetic Organic Chemistry, 21:5, 611-617, DOI:
10.1080/00397919108020827
To link to this article: http://dx.doi.org/10.1080/00397919108020827
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