Bioorganic and Medicinal Chemistry Letters p. 1148 - 1153 (2014)
Update date:2022-08-04
Topics:
Jiang, Jian-Kang
McCoy, Joshua G.
Shen, Min
LeClair, Christopher A.
Huang, Wenwei
Negri, Ana
Li, Jihong
Blue, Robert
Harrington, Amanda Weil
Naini, Sarasija
David III, George
Choi, Won-Seok
Volpi, Elisabetta
Fernandez, Joseph
Babayeva, Mariana
Nedelman, Mark A.
Filizola, Marta
Coller, Barry S.
Thomas, Craig J.
A collection of αIIbβ3 integrin receptor antagonists possessing a unique MIDAS metal ion displacement mechanism of action is presented. Insight into these agents' structure-activity relationships, binding modality, and pharmacokinetic and pharmacodynamic
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