STEREOSELECTIVE ONE-POT SYNTHESES OF TRANS-3-AMINO-β-LACTAMS FROM ZINC ENOLATES OF N-PROTECTED α-AMINOACID ESTERS AND IMINES

DOI: 10.1016/S0040-4039(00)87909-5

Source and publish data:

Tetrahedron Letters p. 2467 - 2470 (1988)

Update date:2022-09-26

Topics:

Authors:

Steen, Fred H. van der

Jastrzebski, Johann T.B.H.

Koten, Gerard van

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0040-4039(00)87909-5

A new one-pot synthesis of 3-amino-β-lactams that is based on the condensation of simple imines with zinc enolates of disilyl protected glycine esters is reported.Isolated yields are high and a trans-selectivity is observed.

Full text of DOI:10.1016/S0040-4039(00)87909-5

Products guided by the article

Product name:3-(2,2,5,5-tetramethyl-1-aza-2,5-disilacyclopentyl)-4-phenyl-2-azetidinone

Cas No:136491-27-5

R&D Labs maybe for 136491-27-5

Zhengzhou HQ Material Co.,Ltd

Contact:+86-371-67759225

Address:No.32, Jinsuo Road, High-tech Zone
Jinhua Haoyuan Chemical CO., LTD(expird)

Contact:86-579-82465583

Address:Jinhua,Zhejiang
NanJing Rate Biochemicals CO., LTD

Contact:+86-25-84931986

Address:NO. 1 Hongjing Road,Jiangning Science Park,Nanjing,China
Shandong Jincheng Zhonghua Bio-pharmaceutical Co.,Ltd

Contact:+86-533-5415882

Address:Zichuan Economic Development Zone,Zibo City,Shandong Province,China
Chengdu Gelipu Biotechnology Co., Ltd.

website:http://www.glp-china.com

Contact:86-28-82610909

Address:chegndu

Relevant to this article

Oxime esters as acylating agents in the aminolysis reaction. A simple and chemoselective method for the preparation of amides from amino alcohols

Doi:10.1055/s-1991-26553
(1991)
Cholesterol modified OPE functionalized film: Fabrication, fluorescence behavior and sensing performance

Doi:10.1039/c2jm16637b
(2012)
Anticancer activity of self-assembled molecular rectangles via arene-ruthenium acceptors and a new unsymmetrical amide ligand

Doi:10.1021/om2012826
(2012)
Silylboranes as new sources of silyl radicals for chain-transfer reactions

Doi:10.1002/chem.201102318
(2012)
Synthesis of 2-anilinopyridine dimers as microtubule targeting and apoptosis inducing agents

Doi:10.1016/j.bmc.2014.11.001
(2014)
(Dynamic) Kinetic Resolution of Enamines/Imines: Enantioselective N-Heterocyclic Carbene Catalyzed [3+3] Annulation of Bromoenals and Enamines/Imines

Doi:10.1002/anie.201813047
(2019)

Article Doi