STEREOSELECTIVE ONE-POT SYNTHESES OF TRANS-3-AMINO-β-LACTAMS FROM ZINC ENOLATES OF N-PROTECTED α-AMINOACID ESTERS AND IMINES

DOI: 10.1016/S0040-4039(00)87909-5

Source and publish data:

Tetrahedron Letters p. 2467 - 2470 (1988)

Update date:2022-09-26

Topics:

Authors:

Steen, Fred H. van der

Jastrzebski, Johann T.B.H.

Koten, Gerard van

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0040-4039(00)87909-5

A new one-pot synthesis of 3-amino-β-lactams that is based on the condensation of simple imines with zinc enolates of disilyl protected glycine esters is reported.Isolated yields are high and a trans-selectivity is observed.

Full text of DOI:10.1016/S0040-4039(00)87909-5

Products guided by the article

Product name:3-(2,2,5,5-tetramethyl-1-aza-2,5-disilacyclopentyl)-4-phenyl-2-azetidinone

Cas No:136491-27-5

R&D Labs maybe for 136491-27-5

Beijing Tianjia Chemical Science & Technology Co.,Ltd

Contact:86-0550-2392698

Address:No.388, Shiliang Road (East),
Hefei TNJ chemical industry co.,ltd

website:https://www.tnjchem.com

Contact:+86-551-65418695

Address:B911 Xincheng Business Center, Qianshan Road, Hefei Anhui China
Jiangsu Wanlong Chemical Co., Ltd.

website:http://www.wanlongchem.com

Contact:+86-511-86810993 0086-511-8681 0888;

Address:Quanzhou Town, Danyang City, Jiangsu
Changzhou BaoKang Pharmaceutical & Chemical Co., Ltd

Contact:(86) 519-88782201 88784080 88785278

Address:Henglin town, changzhou,Jiangsu
Accendatech Co., LTD

Contact:+86-22-83718541

Address:32th Floor, Rongqiao Center Intersection of Changjiang Road and Nankai Six Road Nankai District Tianjin 300102, China

Relevant to this article

Oxime esters as acylating agents in the aminolysis reaction. A simple and chemoselective method for the preparation of amides from amino alcohols

Doi:10.1055/s-1991-26553
(1991)
Cholesterol modified OPE functionalized film: Fabrication, fluorescence behavior and sensing performance

Doi:10.1039/c2jm16637b
(2012)
Anticancer activity of self-assembled molecular rectangles via arene-ruthenium acceptors and a new unsymmetrical amide ligand

Doi:10.1021/om2012826
(2012)
Silylboranes as new sources of silyl radicals for chain-transfer reactions

Doi:10.1002/chem.201102318
(2012)
Synthesis of 2-anilinopyridine dimers as microtubule targeting and apoptosis inducing agents

Doi:10.1016/j.bmc.2014.11.001
(2014)
(Dynamic) Kinetic Resolution of Enamines/Imines: Enantioselective N-Heterocyclic Carbene Catalyzed [3+3] Annulation of Bromoenals and Enamines/Imines

Doi:10.1002/anie.201813047
(2019)

Article Doi