Sequential Addition of 2-Potassio-2-nitropropane and Oxygen to 4-Arylidene-oxazol-5-ones: A New Method for 2-Aryl Butenoic Acid Imides

DOI: 10.1039/c39910000897

Source and publish data:

Journal of the Chemical Society. Chemical communications p. 897 - 899 (1991)

Update date:2022-09-26

Topics:

Authors:

Lalitha, N.

Bhalerao, U. T.

Iyengar, D. S.

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Article abstract of DOI:10.1039/c39910000897

The regiospecific addition of 2-potassio-2-nitropropane to the 4-arylidene-oxazol-5-ones followed by oxygenation led to 2-arylbutenoic acid imides, the key intermediate for several pharmacodynamic compounds in high yields.

Full text of DOI:10.1039/c39910000897

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