Journal of Medicinal Chemistry p. 423 - 430 (1992)
Update date:2022-08-02
Topics:
Mach
Jackson
Luedtke
Ivins
Molinoff
Ehrenkaufer
Two series of N-substituted spiperone analogues were prepared and evaluated in vitro to measure their affinities for dopamine D2 and serotonin 5-HT2 receptors. Substitution of the amide nitrogen with an alkyl group of five carbon uni
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