Analgesic dipeptide derivatives. 7. 3,7-Diamino-2-hydroxyheptanoic acid (DAHHA) containing dipeptide analogues of the analgesic compound H-Lys- Trp(Nps)-OMe

DOI: 10.1021/jm00083a013

Source and publish data:

Journal of Medicinal Chemistry p. 889 - 895 (1992)

Update date:2022-08-03

Topics:

Authors:

Herranz Herranz

Vinuesa Vinuesa

Perez Perez

Garcia-Lopez

Lopez Lopez

De Ceballos

Del Rio Del Rio

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1021/jm00083a013

A series of diastereomeric dipeptides, analogues of the analgesic compound H-Lys-Trp(Nps)-OMe (2), containing 3,7-diamino-2-hydroxyheptanoic acid (DAHHA) and 2-[(o-nitrophenyl)sulfenyl]tryptophan [Trp(Nps)] has been synthesized. These compounds were teste

Full text of DOI:10.1021/jm00083a013

Products guided by the article

Product name:(S)-2-((2S,3S)-3,7-Bis-benzyloxycarbonylamino-2-hydroxy-heptanoylamino)-3-(1H-indol-3-yl)-propionic acid methyl ester

Cas No:138207-77-9

R&D Labs maybe for 138207-77-9

Shanghai Yuanding Chem. Sci. & Tech. Co., Ltd.

website:http://www.shydtec.com

Contact:86-21-57721279

Address:Science and Technology Park, Songjiang District, Shanghai, China
Shijiazhuang Haitian Amino Acid Co., Ltd.

Contact:+86-311-88908111

Address:Shijiazhuang Hebei province,China
SHANXI XINTIANYUAN PHARMACEUTICAL CO., LTD.

website:http://www.tychemical.com

Contact:0086-358-3521713 3521715

Address:No. 1 Yintong Road, Shanxi Jiaocheng Economic Development Zone, Xiajiaying Town, Jiaocheng County, Lvliang City, Shanxi Province, China
Synchem Pharma Co.,Ltd(expird)

Contact:+0086-21-61984905-1

Address:Building 60,Zimian Park, LongYang industrial Area, 1515Nong，Yuandong Road Fengxian District, Shanghai ,China
SHAANXI FUJIE PHARMACEUTICAL CO.,LTD

website:http://www.fujiepharm.com

Contact:+86-29-63650906

Address:Yuanqu Yi Road, Qinghe Food Industrial Park, Sanyuan County, Shaanxi Province, China

Relevant to this article

Al-NiCl(2°)6H₂O-THF: A new, mild and neutral system for selective reduction of organic functional groups

Doi:10.1016/S0040-4020(01)82402-9
(1991)
Enantioselective synthesis of (+)-gossonorol and related systems using organozinc reagents

Doi:10.1016/j.tetasy.2012.04.003
(2012)
Synthesis and antioxidant evaluation of isochroman-derivatives of hydroxytyrosol: Structure-activity relationship

Doi:10.1016/j.foodchem.2014.10.036
(2015)
Discovery, Optimization, and Biological Characterization of 2,3,6-Trisubstituted Pyridine-Containing M₄ Positive Allosteric Modulators

Doi:10.1002/cmdc.201900088
(2019)
DETERMINATION OF THE GEOMETRIC CONFIGURATION OF THE POLYENE CHAIN OF MONO-CIS C₄₀ CAROTENOIDS II A 13C NMR STUDY OF MONO-CIS LUTEINS AND MONO-CIS CAPSANTHINS

Doi:10.1016/S0040-4020(01)97736-1
(1981)
Anti-tumour active gold(i), palladium(ii) and ruthenium(ii) complexes with thio- and selenoureato ligands: A comparative study

Doi:10.1039/c7dt04180b
(2018)

Article Doi