Analgesic dipeptide derivatives. 7. 3,7-Diamino-2-hydroxyheptanoic acid (DAHHA) containing dipeptide analogues of the analgesic compound H-Lys- Trp(Nps)-OMe

DOI: 10.1021/jm00083a013

Source and publish data:

Journal of Medicinal Chemistry p. 889 - 895 (1992)

Update date:2022-08-03

Topics:

Authors:

Herranz Herranz

Vinuesa Vinuesa

Perez Perez

Garcia-Lopez

Lopez Lopez

De Ceballos

Del Rio Del Rio

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Article abstract of DOI:10.1021/jm00083a013

A series of diastereomeric dipeptides, analogues of the analgesic compound H-Lys-Trp(Nps)-OMe (2), containing 3,7-diamino-2-hydroxyheptanoic acid (DAHHA) and 2-[(o-nitrophenyl)sulfenyl]tryptophan [Trp(Nps)] has been synthesized. These compounds were teste

Full text of DOI:10.1021/jm00083a013

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