Decreased histamine release by luteinizing hormone-releasing hormone antagonists obtained upon translocation of the cationic amino acid from position 8 to position 7

DOI: 10.1021/jm00082a004

Source and publish data:

Journal of Medicinal Chemistry p. 636 - 640 (1992)

Update date:2022-08-04

Topics:

Authors:

Flouret Flouret

Mahan Mahan

Majewski

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Article abstract of DOI:10.1021/jm00082a004

We report analogues of N-Ac-D-Nal-D-Cpa-D-Pal-Ser-Lys(Pic)-D-Lys(Pic)-Leu- Ilys-Pro-D-Ala-NH₂, the parent antagonist (PA), which is a potent antagonist of LHRH. To simplify future radioactive labeling we prepared N-Ac-D-Nal-D- Cpa-D-Pal-Ser-Lys

Full text of DOI:10.1021/jm00082a004

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Product name:N-Ac-D-Nal-D-Cpa-D-Pal-Ser-Lys(Pic)-D-Lys(Pic)-Leu-Trp-Pro-D-Arg-NH₂

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