Bioorganic and Medicinal Chemistry p. 1029 - 1039 (2014)
Update date:2022-07-29
Topics: Inhibitors Warburg Effect 6-phosphofructo-2-kinase/2,6-bisphosphatase 3 (PFKFB3) 2-arylpyridazinones Relationships
Brooke, Darby G.
Van Dam, Ellen M.
Watts, Colin K.W.
Khoury, Amanda
Dziadek, Marie A.
Brooks, Hilary
Graham, Lisa-Jane K.
Flanagan, Jack U.
Denny, William A.
High-throughput screening of a small-molecule library identified a 5-triazolo-2-arylpyridazinone as a novel inhibitor of the important glycolytic enzyme 6-phosphofructo-2-kinase/2,6-bisphosphatase 3 (PFKFB3) Such inhibitors are of interest due to PFKFB3's
View MoreKunshan Yalong Trading Co,.Ltd
Contact:86-512-57621185
Address:805-807 Room Hongqiao Mansion ,1088 West Qianjin Road, Kunshan, Jiangsu,China
Contact:+33-5-34012600
Address:28 ZA des Pignès
Ji'nan Orgachem Pharmaceutical Co.,Ltd
Contact:+86-531-82687810
Address:Jinan
Anhui Eapearl Chemical Co., Ltd.
Contact:86-562-5858458
Address:358 South Huaihe Road
ShangHai Ruiyi Medical Technology Co.,Ltd.
Contact:+86-21-54718086
Address:No951 Jianchuan RD,Minhang District
Doi:10.1016/S0040-4020(01)82175-X
(1966)Doi:10.1021/ic301691d
(2012)Doi:10.1016/j.tetlet.2012.09.051
(2012)Doi:10.1039/c39920000549
(1992)Doi:10.1016/j.tetlet.2012.09.114
(2012)Doi:10.1021/jm301345v
(2012)