Development of N-[4-[6-(isopropylamino)pyrimidin-4-yl]-1,3-thiazol-2-yl]-N -methyl-4-[11C]methylbenzamide for positron emission tomography imaging of metabotropic glutamate 1 receptor in monkey brain

DOI: 10.1021/jm301597s

Source and publish data:

Journal of Medicinal Chemistry p. 11042 - 11051 (2012)

Update date:2022-09-26

Topics:

Authors:

Fujinaga, Masayuki

Yamasaki, Tomoteru

Maeda, Jun

Yui, Joji

Xie, Lin

Nagai, Yuji

Nengaki, Nobuki

Hatori, Akiko

Kumata, Katsushi

Kawamura, Kazunori

Zhang, Ming-Rong

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Article abstract of DOI:10.1021/jm301597s

Three novel 4-substituted benzamides have been synthesized as potential ligands for the positron emission tomography (PET) imaging of metabotropic glutamate 1 (mGlu1) receptor in the brain. Of these compounds, N-(4-(6-(isopropylamino)pyrimidin-4-yl)-1,3-t

Full text of DOI:10.1021/jm301597s

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Product name:N-[4-(6-chloropyrimidin-4-yl)-1,3-thiazol-2-yl]-N,4-dimethylbenzamide

Cas No:1414953-54-0

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Wuxi Morality Chemical Co., Ltd(expird)

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