Anti-inflammatory phospholipase-A2 inhibitors. II. Design, synthesis and structure-activity relationship

DOI: 10.1016/0223-5234(92)90138-Q

Source and publish data:

European Journal of Medicinal Chemistry p. 595 - 610 (1992)

Update date:2022-09-26

Topics:

Authors:

Wilkerson

DeLucca DeLucca

Galbraith

Kerr Kerr

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Article abstract of DOI:10.1016/0223-5234(92)90138-Q

The design and synthesis of a novel series of phospholipase-A₂ (PLA₂) inhibitor with antiinflammatory activity was based on a systematic structure-activity relationship (SAR) analysis.

Full text of DOI:10.1016/0223-5234(92)90138-Q

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