Novel benzamides as selective and potent gastrokinetic agents. IV. Synthesis and structure-activity relationships of 2-substituted 4-amino-N-[(4-benzyl-2-morpholinyl)methyl]-5-chlorobenzamides

DOI: 10.1248/cpb.40.1470

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 1470 - 1475 (1992)

Update date:2022-08-04

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Authors:

Kato Kato

Morie Morie

Yoshida Yoshida

Matsumoto

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Article abstract of DOI:10.1248/cpb.40.1470

A new series of 2-substituted 4-amino-N-[(4-benzyl-2-morpholinyl)methyl]-5-chlorobenzamides (4-39) including a few 4-fluorobenzyl analogues were prepared and evaluated for their gastrokinetic activity by determining their effects on the gastric emptying a

Full text of DOI:10.1248/cpb.40.1470

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Product name:4-Amino-N-(4-benzyl-morpholin-2-ylmethyl)-5-chloro-2-propoxy-benzamide

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