Protection of primary amino as pyrrole in organometallic reagents

DOI: 10.1016/S0040-4039(00)74737-X

Source and publish data:

Tetrahedron Letters p. 8125 - 8126 (1992)

Update date:2022-09-26

Topics:

Authors:

Davis Davis

Egan Egan

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Article abstract of DOI:10.1016/S0040-4039(00)74737-X

Pyrrole 5 was converted into Grignard and organocuprate reagents. After addition of the latter to alkene 6, the pyrrole ring was converted to a primary amine by ozonolysis, reduction and hydrolysis.

Full text of DOI:10.1016/S0040-4039(00)74737-X

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