Bioorganic and Medicinal Chemistry Letters p. 177 - 180 (2014)
Update date:2022-09-26
Topics:
Schroder, Tenna Juul
Christensen, Soren
Lindberg, Samsa
Langgard, Morten
David, Laurent
Maltas, Philip J.
Eskildsen, Jorgen
Jacobsen, Jan
Tagmose, Lena
Simonsen, Klaus Baek
Biilmann Ronn, Lars Christian
De Jong, Inge E.M.
Malik, Ibrahim J.
Karlsson, Jens-Jakob
Bundgaard, Christoffer
Egebjerg, Jan
Stavenhagen, Jeffrey B.
Strandbygard, Dorthe
Thirup, Soren
Andersen, Jacob Lauwring
Uppalanchi, Srinivas
Pervaram, Sridhar
Kasturi, Shiva Prasad
Eradi, Pradheep
Sakumudi, Durga Rao
Watson, Stephen P.
The identification of the novel, selective, orally bioavailable Sortilin inhibitor AF38469 is described. Structure-activity relationships and syntheses are reported, along with an X-ray crystal structure of the sortilin-AF38469 protein-inhibitor complex.
View MoreFREEBARQUE DEVELOPMENT GROUP LIMITED
Contact:+86(0)10-5109 5335 or 5109 5345
Address:Room602,Block1-B,LINGDI OFFICE,NO.13 BEIYUAN ROAD
Henan zhongda Biological Engineering Co., Ltd
Contact:86-28-18109029985
Address:shenzhou road,xuedian industrial estate,zhengzhou city,henan province CHN
HUNAN CHEMAPI BIOLOGICAL TECHNOLOGY CO.,LTD.
Contact:+86-186-02659358
Address:1004, building 3, Wanke Jinsemaitianyuan, 498 Guitang Road, Yuhua District, Changsha City, Hunan Province, China
Shanghai Balmxy Pharmaceutical Co., Ltd
Contact:0086-21-24206007
Address:Room 402, 15#, No. 909 wangyue Road, shanghai, P. R. China
Nanjing Fubang Chemical Co.,Ltd
Contact:+86-25-83179199
Address:5F,Tianzheng international plaza,No399 Zhongyang Road ,Nanjing China
Doi:10.1021/jo00115a003
(1995)Doi:10.1055/s-2007-965919
(2007)Doi:10.1128/AAC.03958-14
(2015)Doi:10.1246/bcsj.66.2936
(1993)Doi:10.1016/S0040-4020(01)81811-1
(1993)Doi:10.1016/S0040-4039(00)95278-X
(1989)