European Journal of Medicinal Chemistry p. 95 - 105 (1994)
Update date:2022-08-03
Topics:
Colotta
Cecchi
Catarzi
Filacchioni
Galli
Mori
The synthesis and in vitro GABA(A) activity as GABA(A) antagonists of some 1-aminophthalazinium salts and imidazophthalazines are reported. Structure-activity relationships and a molecular modelling study allowed us to define the features which determine
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