Journal of Medicinal Chemistry p. 7449 - 7464 (2015)
Update date:2022-08-15
Topics:
Damont, Annelaure
Médran-Navarrete, Vincent
Cacheux, Fanny
Kuhnast, Bertrand
Pottier, Géraldine
Bernards, Nicholas
Marguet, Frank
Puech, Frédéric
Boisgard, Rapha?l
Dollé, Frédéric
A series of novel pyrazolo[1,5-a]pyrimidines, closely related to N,N-diethyl-2-(2-(4-(2-fluoroethoxy)phenyl)-5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)acetamide (2, DPA-714), were synthesized and biologically in vitro evaluated for their potential to bind
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