Journal of Medicinal Chemistry p. 8369 - 8384 (2017)
Update date:2022-08-15
Topics:
McDaniel, Keith F.
Wang, Le
Soltwedel, Todd
Fidanze, Steven D.
Hasvold, Lisa A.
Liu, Dachun
Mantei, Robert A.
Pratt, John K.
Sheppard, George S.
Bui, Mai H.
Faivre, Emily J.
Huang, Xiaoli
Li, Leiming
Lin, Xiaoyu
Wang, Rongqi
Warder, Scott E.
Wilcox, Denise
Albert, Daniel H.
Magoc, Terrance J.
Rajaraman, Ganesh
Park, Chang H.
Hutchins, Charles W.
Shen, Jianwei J.
Edalji, Rohinton P.
Sun, Chaohong C.
Martin, Ruth
Gao, Wenqing
Wong, Shekman
Fang, Guowei
Elmore, Steven W.
Shen, Yu
Kati, Warren M.
The development of bromodomain and extraterminal domain (BET) bromodomain inhibitors and their examination in clinical studies, particularly in oncology settings, has garnered substantial recent interest. An effort to generate novel BET bromodomain inhibi
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