Enantiomerically pure amino alcohols and diamino alcohols from L-aspartic acid. Application to the synthesis of epi- and diepislaframine

DOI: 10.1021/jo00101a042

Source and publish data:

Journal of Organic Chemistry p. 6766 - 6776 (1994)

Update date:2022-09-26

Topics:

Authors:

Gmeiner Gmeiner

Junge Junge

Kartner Kartner

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Article abstract of DOI:10.1021/jo00101a042

Starting from natural aspartic acid (6) a practical method for the synthesis of enantiomerically pure 3-amino alcohols 8 including 3,4-diamino derivatives is described. After perbenzylation of 6 and reduction of both carboxylates, position 4 of the result

Full text of DOI:10.1021/jo00101a042

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