
Journal of Heterocyclic Chemistry p. 1171 - 1176 (1994)
Update date:2022-08-05
Topics:
Gatta
Del Giudice
Borioni
Mustazza
Fazio
This paper describes the preparation of 2-aryl-8-fluorobenzyl-1,2,4-triazolo[5,1-i]purines 2, starting from 2-aryl-7,8-diamino-1,2,4-triazolo[1,5-c]pyrimidines 9. Our synthetic procedure represents the first example of a feasible approach for the synthesi
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