Full functionalization of the imidazole scaffold by selective metalation and sulfoxide/magnesium exchange

DOI: 10.1002/anie.201309217

Source and publish data:

Angewandte Chemie - International Edition p. 1430 - 1434 (2014)

Update date:2022-07-30

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Authors:

Samann, Christoph

Coya, Estibaliz

Knochel, Paul

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Article abstract of DOI:10.1002/anie.201309217

A simple, flexible, and straightforward method for the functionalization of all the positions of the imidazole heterocycle through regioselective arylations, allylations, acylations, and additions to aldehydes is disclosed. Starting from the readily avail

Full text of DOI:10.1002/anie.201309217

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